Anastrozole

GENETIC PHARMACEUTICALS ANASTROZOLE

Anastrozole, containing the active substance Anastrozole 1 mg, is a potent aromatase inhibitor designed to counteract estrogen-related issues in medical and bodybuilding contexts.

DRUG COMPOSITION

Each Anastrozole tablet comprises precisely 1 mg of Anastrozole, ensuring accuracy in dosing.

PHARMACEUTICAL FORM

Anastrozole is available in oral tablet form, providing a convenient means of administration.

PHARMACEUTICAL GROUP AND ATC CODE

As an aromatase inhibitor, Anastrozole belongs to the group of antineoplastic and immunomodulating agents. Its Anatomical Therapeutic Chemical (ATC) code is L02BG03.

PHARMACOLOGICAL PROPERTIES

Anastrozole inhibits aromatase, the enzyme responsible for estrogen synthesis, effectively lowering estrogen levels. This property makes it valuable in treating estrogen-dependent conditions and preventing estrogenic side effects.

PROFILE

• Chemical name: 2,2'-[5-(1H-1,2,4-triazol-1-ylmethyl)-1,3-phenylene]bis(2-methylpropanenitrile)
• Chemical formula: C17H19N5
• Percentage of anabolic activity: Not a steroid
• Percentage of androgenic activity: Not a steroid
• Active half life: Approximately 46 hours
• Recommended dosage: 1 mg per day for breast cancer; may vary in other applications
• Acne: Not reported
• Bloating (water retention): Not reported
• HBR: Low
• Hepatic toxicity: Rare
• Aromatization: Inhibits aromatase, reducing estrogen conversion

THERAPEUTICAL INDICATIONS

Anastrozole is indicated for the treatment of hormone receptor-positive breast cancer. In bodybuilding, it is employed to mitigate estrogenic side effects resulting from anabolic steroid use.

DOSES AND METHOD OF ADMINISTRATION

For men in bodybuilding, the recommended Anastrozole dose typically ranges from 0.25 to 1 mg every other day or 0.5 mg every third day. Women usually require lower doses, if necessary, due to the potential for estrogen suppression.

CYCLE/STACKING

Solo Cycle:

• Start with 0.25 mg every other day, adjusting as needed based on estrogen response. Cycle lengths can vary but are often aligned with the duration of anabolic steroid use.

Cutting Cycle:

• Combine Anastrozole with compounds prone to aromatization, such as Testosterone. Example: Anastrozole 0.5 mg every other day with Testosterone Propionate 100 mg every other day for an 8-week cutting cycle.

Bulking Cycle:

• Include Anastrozole in bulking cycles where aromatizable compounds like Deca are used. Example: Anastrozole 1 mg every other day with Nandrolone Decanoate 400 mg per week for a 12-week bulking cycle.

POST CYCLE THERAPY

Anastrozole is not typically utilized in post-cycle therapy (PCT) as its use revolves around preventing estrogenic issues during the cycle. PCT commonly involves substances like SERMs (Selective Estrogen Receptor Modulators).

SIDE EFFECTS

Possible side effects include joint pain, fatigue, and osteoporosis. Dosing should be monitored to prevent excessive estrogen suppression.

CONTRAINDICATIONS

Individuals with known hypersensitivity to Anastrozole or experiencing severe osteoporosis should avoid its use.

OVERDOSE

In case of overdose symptoms, seek medical attention promptly. No specific antidote is known.

WARNINGS AND SPECIAL PRECAUTIONS FOR USE:

Regular bone density assessments are recommended for individuals on prolonged Anastrozole treatment due to potential bone health implications.

INTERACTIONS WITH OTHER DRUGS

Exercise caution when combining Anastrozole with other drugs, particularly those affecting liver function or bone health.

PRESENTATION, PACKAGING

1 mg per tablet, 50 tablets in sachet.

STORAGE

Store Anastrozole in a cool, dry place, away from direct sunlight and moisture. Keep it out of reach of children.

DELIVERY TO THE USA

Our delivery services ensure Anastrozole reaches customers in the USA safely and efficiently.

LEGAL STATUS

Anastrozole is subject to regulatory restrictions, and its purchase and use should adhere to local laws and regulations. Verify the legal status before obtaining Anastrozole.

DATE OF LAST TEXT CHECKS

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NAME AND ADDRESS OF THE MANUFACTURER

Genetic Pharmaceuticals
India

EXTERNAL LINKS

• Anastrozole Wiki, wikipedia.org
• Anastrozole Uses, Side Effects & Warnings, drugs.com
• Anastrozole Oral: Uses, Side Effects, Interactions, Pictures, webmd.com.